I-250mg triclabendindale bos

Inkcazo emfutshane:

Imbonakalo:I-bolus emhlophe

I-bos ubunzima:I-0.5g ~ 19g

Izenzo kunye nokusetyenziswa:I-Bebimididabole Anti-Fasciola ichiza. Isetyenziselwa ikakhulu ukuthintela kunye nonyango lwe-Fasciola Hepatica Hepatica kwiinkomo kunye neegusha.

Izatifikethi:I-GMP kunye ne-ISO

Isampulu:Iyafumaneka

Beka ubomi kwishelufa:3years

 

 


Ixabiso le-fob I-US $ 0.5 - 9,999 / isiqwenga
Imiz.Order I-1 iqhekeza
Amandla obonelelo I-10000 yeziqwenga ngenyanga
Ithuba lokuhlawula T / t, d / p, d / a, l / c
iinkamela iinkomo iibhokhwe iigusha

Iinkcukacha zemveliso

Iprofayile yekhampani

Iimpawu zeMveliso

Izenzo ze-Pharmacological

I-pharmacodynamics triclobendiolle yeyakwiklasi ye-BezimiDaole ye-BezimiDaole yeziyobisi, isetyenziselwa ukuphepha i-Fasciola Hepatica, kwaye inesiphumo esibonakalayo se-Fasciola Hepatica yeminyaka eyahlukeneyo. amayeza okufihla. Emva kokuba ichiza lithathwe, liphazamisane nesakhiwo se microtubule kunye nomsebenzi weparasite, thintela ukukhululwa kwe-ratiolytic ye-hydrolytic ye-hydrolytic. Iziphumo zeTriclobendindale kwiimpethu ziyahluka ngokuxinana, njengabadala ngendlela ephantsi (1 ~ 4μg / ml)

Ichiza lisaqhubeka lisinda kwiiyure ezingama-24, kwaye umsebenzi uqhekeke kakhulu kwixinzelelo oluphezulu (10-25μg / ml) iiyure ezingama-24; Ukugxininisa okuphezulu kwe-25-50μg / ml ithobela ngokupheleleyo iiyure ezingama-24. Kodwa inovelwano ngakumbi kwiimpethu. Ngo-10 μg / ml, yonke imisebenzi engama-24 yathintelwa.

I-pharmacokinetics

I-biaaaifFument ye-triclobendindale iphezulu. Emva kolawulo lomlomo lwe-10 mg / kg ubunzima bomzimba kunye neegusha, iyeza le-Plaak, iyeza le-Peak lifikelela kwi-15 μ ukuya kwiiyure ezingama-24 ukuya kwengama-36 kwiiyure ezingama-24 ukuya kwi-metabolites ye-tricaboble kunye ne-metabolites zayo. Ixabiso lencopho lechiza lingamaxesha ama-5 ukuya kwangama-20 ukuba kwelinye i-antimisidalisole, kunye nokupheliswa kwesiqingatha sobomi malunga neeyure ezingama-22. I-Triclobendale iyoyinyaziswa kakhulu kwigusha nakwiigundane kwi-Sulfone kunye neSulfotisides, ebophelela kwi-albhamun kwaye iqhubeka kwiPlasma ngaphezulu kweentsuku ezisi-7. Ukugxininiswa kweplasma ephezulu kunye nokubopha kwi-plasma albinto kubonakala ngathi kunxulunyaniswa nexesha elide lesenzo se-antifascioli. Emva kweentsuku ezili-10 zolawulo lweziyobisi kwiigusha, malunga ne-95% yechiza ikhutshiwe kwimithombo, i-2% ikhutshiwe kumchamo, kwaye ngaphantsi kwe-1% ikhutshiwe kubisi.

Triclabendindale boslus 250mg

Izenzo kunye nokusetyenziswa

I-Bebimididabole Anti-Fasciola ichiza. Isetyenziselwa ikakhulu ukuthintela kunye nonyango lwe-Fasciola Hepatica Hepatica kwiinkomo kunye neegusha.

Impendulo embi

AKUKHO BUNGOZI OLUFANELEKILEYO KUFUNEKA LONTO XA KUSETYENZISELWA NGOKUSETYENZISELWEYO NGOKUSETYENZISWA KOMNYANGO NOKUFUNDA

Ukulumkela

(1) Ukhubazekile ngexesha lemveliso yobisi.

(2) Inetyhefu kakhulu kwiintlanzi, kwaye isikhongozelo seziyobisi esiseleyo akufuneki singcolise umthombo wamanzi.

.

(4) Hlamba izandla emva kokufaka isicelo

Ixesha lokurhoxa

Iintsuku ezingama-56 zeenkomo kunye neegusha

Ukugcinwa

Ivenkile kule ndawo ingezantsi kwe-30 ℃.


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    I-Hebei Veyolong Pharmaceutical Co., i-LTD, ibekwe kwiSixeko saseShijiazhuang, kwiPhondo laseHebei, iChina, ecaleni kwengxowa ye-Beijing. Uyishishini elikhulu eliqinisekisiweyo le-GMP le-GEMP ye-GEMP, ene-R & D, ukuvelisa kunye nentengiso ye-Veterinal Apis, amalungiselelo, i-PREPEDED yezongezo. Njengeziko lobugcisa lePhondo, iVeyong iseke inkqubo ye-R & D yeS System yeZiyobisi eziNtsha zeZilwanyana, kwaye zisekelezwe kwishishini lezonyango lwezilwanyana, kukho iingcali ezingama-65 zezobugcisa. IVeyong ineziseko zambini zemveliso: Shijiazhuang kunye ne-Shijiazduang Isiseko esinendawo ye-78,706 M2, i-APPINECTINE YEMIQATHANGO YOKUGQIBELA, I-APIALITINE YOKUGQIBELA I-IYIMATION, i-APIALITCINE YEMIQATHANGO YOKUGQIBELA, INDAWO YOKUGQIBELA, I-PREPE, Izitshabalalisi kunye nentsholongwane, i-ECT. IVeyong ibonelela nge-APIs, amalungiselelo angaphezu kwe-100 yeelebheli, kunye nenkonzo ye-OEM ye-ODM.

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